Found 1 Enz. Inhib. hit(s) with Target = 'Bifunctional phosphoribosylaminoimidazole carboxylase/phosphoribosylaminoimidazole succinocarboxamide synthetase' and Ligand = 'BDBM489214'
TargetBifunctional phosphoribosylaminoimidazole carboxylase/phosphoribosylaminoimidazole succinocarboxamide synthetase(Human)
Lifearc
US Patent
Lifearc
US Patent
Affinity DataIC50: <10nMAssay Description:5 μl WT full length PAICS (final assay concentration, fac, 2.5 nM) in basic buffer, added to black, non-binding, 384-well plates (Corning #3575)...More data for this Ligand-Target Pair