Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Breast cancer type 1 susceptibility protein' and Ligand = 'BDBM50345640'
TargetBreast cancer type 1 susceptibility protein(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345640((S)-2-((2S,3R)-2-((S)-1-((S)-2-acetamido-3-(phosph...)
Affinity DataKd:  190nMAssay Description:Binding affinity to BRCA1 by isothermal titration calorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetBreast cancer type 1 susceptibility protein(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345640((S)-2-((2S,3R)-2-((S)-1-((S)-2-acetamido-3-(phosph...)
Affinity DataKi:  270nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBreast cancer type 1 susceptibility protein(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345640((S)-2-((2S,3R)-2-((S)-1-((S)-2-acetamido-3-(phosph...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed