Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Broad substrate specificity ATP-binding cassette transporter ABCG2' and Ligand = 'BDBM50370873'
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5086 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50370873(CHEMBL222265)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of BCRP expressed in human HEK293 cells assessed as maximal mitoxantrone accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed