Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Bromodomain and PHD finger-containing protein 3' and Ligand = 'BDBM50249810'
TargetBromodomain and PHD finger-containing protein 3(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50249810(CHEMBL4102050)
Affinity DataIC50:  260nMAssay Description:Inhibition of human BRPF3 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain and PHD finger-containing protein 3(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50249810(CHEMBL4102050)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human His tagged BRPF3 incubated for 30 mins followed by addition of biotinylated peptide and further incubation for 30 mins measured b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain and PHD finger-containing protein 3(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50249810(CHEMBL4102050)
Affinity DataKd:  940nMAssay Description:Binding affinity to human BRPF3 by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed