Report error Found 28 Enz. Inhib. hit(s) with Target = 'Bromodomain testis-specific protein' and Ligand = 'BDBM50365262'
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataKd: 190nMAssay Description:Binding affinity to BRDT-BD1 by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataKd: 183nMAssay Description:Binding affinity to recombinant BRDT BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataKd: 217nMAssay Description:Binding affinity to recombinant BRDT BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataKd: 260nMAssay Description:Binding affinity to recombinant human N-terminal hexaHis-tagged BRDT expressed in Escherichia coli BL21 (DE3) cells by MST assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataKd: 22nMAssay Description:Binding affinity to recombinant human N-terminal hexaHis-tagged BRDT expressed in Escherichia coli BL21 (DE3) cells by qPCR assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataKd: 188nMAssay Description:Binding affinity to recombinant human N-terminal hexaHis-tagged BRDT expressed in Escherichia coli BL21 (DE3) cells by ITC analysisMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataKd: 188nMAssay Description:Binding affinity to his tagged BRDT bromodomain (unknown origin) assessed as dissociation constant by SPR methodMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Binding affinity to human partial length BRDT BD2 (K250 to E382 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotin...More data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of BRDT (unknown origin)More data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 77nMAssay Description:ssays were performed as described previously with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were dilu...More data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 103nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 103nMAssay Description:Binding affinity to BRDT bromodomain (unknown origin) by alpha screen assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of BRDT D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 124nMAssay Description:Binding affinity to BRDT bromodomain (unknown origin) by alpha screen assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 134nMAssay Description:Inhibition of BRDT bromodomain 1 (unknown origin) by Alphascreen based methodMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 134nMAssay Description:Inhibition of human recombinant His-tagged BRDT BD1 domain expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells by AlphaScreen assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 147nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150 mM ...More data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 178nMAssay Description:Binding affinity BRDT BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 183nMAssay Description:Inhibition of BRDT BD1 (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 185nMAssay Description:Inhibition of BRDT BD2 (unknown origin) incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 207nMAssay Description:Inhibition of BRDT BD1 (unknown origin) incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 217nMAssay Description:Inhibition of BRDT BD2 (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 224nMAssay Description:Binding affinity BRDT BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 325nMAssay Description:Inhibition of recombinant BRDT BD2 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Binding affinity to human partial length BRDT BD1 (N21 to E137 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 534nMAssay Description:Inhibition of recombinant BRDT BD1 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Human)
Japan Science and Technology Agency
Curated by ChEMBL
Japan Science and Technology Agency
Curated by ChEMBL
Affinity DataIC50: 588nMAssay Description:Inhibition of recombinant BRDT BD1 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
