Found 3 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 1' and Ligand = 'BDBM50249810' TargetBromodomain-containing protein 1(Homo sapiens (Human))
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibition of human BRPF2-BRD1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 1(Homo sapiens (Human))
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 760nMAssay Description:Inhibition of human His tagged BRPF2 incubated for 30 mins followed by addition of biotinylated peptide and further incubation for 30 mins measured b...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 1(Homo sapiens (Human))
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataKd: 210nMAssay Description:Binding affinity to human BRPF2 by isothermal titration calorimetryMore data for this Ligand-Target Pair
