Found 2 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4' and Ligand = 'BDBM50030894'
Affinity DataIC50: 637nMAssay Description:Inhibition of BRD4 (unknown origin) by biotinylated-JQ1 based AlphaScreen BRD binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 550nMAssay Description:Binding affinity to BRD4 (unknown origin) by isothermal titration colorimetryMore data for this Ligand-Target Pair