Found 1 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4' and Ligand = 'BDBM50458961'
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 107nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair