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Found 1 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4 [49-170]' and Ligand = 'BDBM449845'
TargetBromodomain-containing protein 4 [49-170](Homo sapiens (Human))
Epigenetix

US Patent
LigandPNGBDBM449845(5-[2-cyclopropyl-3-[2-(trifluoromethoxy)ethyl]benz...)
Affinity DataIC50:  190nMAssay Description:To measure activity of bromodomain inhibitors, a His-epitope tagged BRD4 BD149-170 is purchased from BPS Bioscience. BRD4 binding and inhibition is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent