Found 11 Enz. Inhib. hit(s) with Target = 'Butyrophilin subfamily 3 member A1' and Ligand = 'BDBM50236894'
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 2.56E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 3.19E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 W421A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 3.22E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R442A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 3.39E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 M424A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 3.83E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R499A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 3.85E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 3.93E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R448A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: 4.00E+3nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of interleukin 2 stimulated cell proliferation treated for 72 hrs measured...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: 3.40E+3nMAssay Description:Activation of BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of IL2-stimulated IFNgamma production measured after 48 hrs ...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataKd: 1.11E+5nMAssay Description:In vitro for its ability to displace [3H]- spiperone from cloned human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: 4.00E+3nMAssay Description:Activation of BTN3A1 in human PBMC-derived Vgamma9/Vdelta2 T cells assessed as induction of IL2-stimulated cell proliferation by measuring increase i...More data for this Ligand-Target Pair