Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with Target = 'Butyrophilin subfamily 3 member A1' and Ligand = 'BDBM50516696'
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  1.04E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  1.07E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  3.24E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 W421A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  3.43E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R442A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  3.72E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R499A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  4.62E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R448A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  5.35E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 M424A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed