Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'C-X-C chemokine receptor type 4' and Ligand = 'BDBM50196257'
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50196257(CHEMBL3903301)
Affinity DataIC50:  59nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50196257(CHEMBL3903301)
Affinity DataEC50:  52nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed