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Found 3 Enz. Inhib. hit(s) with Target = 'C-X-C chemokine receptor type 4' and Ligand = 'BDBM50603567'
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50603567(CHEMBL5172755)
Affinity DataIC50:  1.60nMAssay Description:Antagonist activity at CXCR4 receptor in SDF-1alpha-stimulated human SUP-T1 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50603567(CHEMBL5172755)
Affinity DataIC50:  12nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells measured by 12G5 competitive binding methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50603567(CHEMBL5172755)
Affinity DataIC50:  236nMAssay Description:Antagonist activity at CXCR4 receptor in human SUP-T1 cells assessed as reduction in SDF-1alpha-stimulated cell migration and measured by CellTiter-9...More data for this Ligand-Target Pair
In DepthDetails PubMed