Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'C-X-C chemokine receptor type 6' and Ligand = 'BDBM50539457'
TargetC-X-C chemokine receptor type 6(Homo sapiens)
Sanford Burnham Prebys Medical Discovery Institute

Curated by ChEMBL
LigandPNGBDBM50539457(CHEMBL4645971)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of CXCL16-induced beta-arrestin recruitment by DiscoveRx cell based...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 6(Homo sapiens)
Sanford Burnham Prebys Medical Discovery Institute

Curated by ChEMBL
LigandPNGBDBM50539457(CHEMBL4645971)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of forskolin-induced cAMP accumulation by DiscoveRx cell based assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 6(Mus musculus)
Sanford Burnham Prebys Medical Discovery Institute

Curated by ChEMBL
LigandPNGBDBM50539457(CHEMBL4645971)
Affinity DataIC50:  1.80E+4nMAssay Description:Antagonist activity at mouse CXCR6 by DiscoveRx cell based beta-arrestin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed