Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Calpain-1 catalytic subunit' and Ligand = 'BDBM50105244'
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50105244(2-Ethyl-1,1-dioxo-1,2,6,7-tetrahydro-5,8-dioxa-1la...)
Affinity DataIC50:  8nMAssay Description:Inhibitory activity towards human calpain IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50105244(2-Ethyl-1,1-dioxo-1,2,6,7-tetrahydro-5,8-dioxa-1la...)
Affinity DataIC50:  8nMAssay Description:In vitro inhibitory activity against recombinant human calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50105244(2-Ethyl-1,1-dioxo-1,2,6,7-tetrahydro-5,8-dioxa-1la...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibitory concentration against MOLT-4 cells (human T-cell leukemia cell line)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed