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Found 2 Enz. Inhib. hit(s) with Target = 'Calpain-1 catalytic subunit' and Ligand = 'BDBM50149195'
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50149195(1-Benzyl-2,3-dihydro-1H-indole-5-carboxylic acid [...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against on human calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50149195(1-Benzyl-2,3-dihydro-1H-indole-5-carboxylic acid [...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against on calpain in C6 glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed