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Found 1 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM29070'
TargetCannabinoid receptor 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM29070(lactam-based compound, 12i)
Affinity DataKi:  0.700nM ΔG°:  -53.1kJ/mole EC50:  0.800nMpH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed