Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50055267'
TargetCannabinoid receptor 1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50055267(CHEMBL3323682)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]CP-55,940 from human recombinant CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50055267(CHEMBL3323682)
Affinity DataEC50:  138nMAssay Description:Agonist activity at human recombinant CB1 receptor expressed in CHO cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed