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Found 4 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50061116'
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50061116(3-(1',1'-dimethylheptyl)-1-hydroxy-9-methyl-6H-ben...)
Affinity DataKi:  33nMAssay Description:Binding to Cannabinoid receptor 1 using African green monkey (COS-7) cells transfected with the cDNA of rat CB1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50061116(3-(1',1'-dimethylheptyl)-1-hydroxy-9-methyl-6H-ben...)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50061116(3-(1',1'-dimethylheptyl)-1-hydroxy-9-methyl-6H-ben...)
Affinity DataKi:  73nMAssay Description:Binding affinity for Cannabinoid receptor 1 using African green monkey (COS-7) cells transfected with the cDNA of rat brain synaptosomal membrane pre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50061116(3-(1',1'-dimethylheptyl)-1-hydroxy-9-methyl-6H-ben...)
Affinity DataEC50:  9.60nMAssay Description:Effective concentration for inhibition of Cannabinoid receptor 1-mediated adenylylcyclase activity using African green monkey (COS-7) cells transfect...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed