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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50408222'
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408222(CHEMBL4174442)
Affinity DataKi:  113nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408222(CHEMBL4174442)
Affinity DataEC50:  182nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cell membranes after 90 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed