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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50603278'
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50603278(CHEMBL5176554)
Affinity DataKi:  0.690nMAssay Description:Displacement of [3H]-CP-55,940 from CB1R in rat brain membranes measured by radioligand based competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50603278(CHEMBL5176554)
Affinity DataEC50:  3.90nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation measured for 60 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed