Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50272395'
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Amgen

Curated by ChEMBL
LigandPNGBDBM50272395(CHEMBL499066 | N-(3-(3-(2-Chloro-4-fluorophenyl)-1...)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at rat recombinant CB2 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated intracellular cAMP levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50272395(CHEMBL499066 | N-(3-(3-(2-Chloro-4-fluorophenyl)-1...)
Affinity DataEC50:  0.0150nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in Sf9 cells by GTP-europium binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50272395(CHEMBL499066 | N-(3-(3-(2-Chloro-4-fluorophenyl)-1...)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated intracellular cAMP levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed