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Found 4 Enz. Inhib. hit(s) with Target = 'Capsid protein' and Ligand = 'BDBM50366817'
TargetCapsid protein(Hepatitis B virus)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50366817(Epivir)
Affinity DataIC50: <100nMAssay Description:Inhibition of capsid protein in Hepatitis B virus infected in human HepG2.2.15 cells assessed as reduction in viral DNA level at 4 uM supplemented wi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid protein(Hepatitis B virus)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50366817(Epivir)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of capsid protein in lamivudine/entecavir-resistant Hepatitis B virus harboring rtL180M/rtM204V/rt184L mutant infected in human HepG2.2.15...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid protein(Hepatitis B virus)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50366817(Epivir)
Affinity DataEC50:  370nMAssay Description:Inhibition of capsid protein in HBV infected in human HepDES19 cells assessed as inhibition of viral replication incubated for 3 days by strand prefe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid protein(Hepatitis B virus)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50366817(Epivir)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of capsid in HBV infected in human HepAD38 cells assessed as reduction in tetracycline-induced cccDNA formation by measuring reduction in ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed