Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Carnitine O-palmitoyltransferase 1, liver isoform' and Ligand = 'BDBM50403044'
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403044BDBM50403044(CHEMBL179241)
Affinity DataEC50:  3.00E+3nMAssay Description:Increase in CPT1 activity in human MCF7 cells assessed as increase in radiolabeled palmitoylcarnitineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403044BDBM50403044(CHEMBL179241)
Affinity DataEC50:  3.00E+3nMAssay Description:Activation of CPT-1 in digitonin-permeabilized human MCF7 cells preincubated for 2 hrs followed by digitonin addition for 6 mins by liquid scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed