Found 4 Enz. Inhib. hit(s) with Target = 'Casein kinase I isoform alpha-like' and Ligand = 'BDBM2579'
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of human CK1a1L using KRRRAL[pS]VASLPGL as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 2.41E+3nMAssay Description:Inhibition of human CK1a1L using KRRRAL[pS]VASLPGL as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 250nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 250nMAssay Description:Binding constant for full-length CSNK1A1LMore data for this Ligand-Target Pair