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Found 4 Enz. Inhib. hit(s) with Target = 'Casein kinase II subunit alpha' and Ligand = 'BDBM165202'
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Senhwa Biosciences

US Patent
LigandPNGBDBM165202(US8168651, Compound TABLE 14A.5 | US9062043, Table...)
Affinity DataIC50:  180nMpH: 7.2Assay Description:Test compounds in aqueous solution were added at a volume of 10 microliters, to a reaction mixture comprising 10 microliters Assay Dilution Buffer (A...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Senhwa Biosciences

US Patent
LigandPNGBDBM165202(US8168651, Compound TABLE 14A.5 | US9062043, Table...)
Affinity DataIC50:  180nMAssay Description:Test compounds in aqueous solution were added at a volume of 10 microliters, to a reaction mixture comprising 10 microliters Assay Dilution Buffer (A...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Senhwa Biosciences

US Patent
LigandPNGBDBM165202(US8168651, Compound TABLE 14A.5 | US9062043, Table...)
Affinity DataKd:  8.90nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Senhwa Biosciences

US Patent
LigandPNGBDBM165202(US8168651, Compound TABLE 14A.5 | US9062043, Table...)
Affinity DataKd:  8.90nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed