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Found 4 Enz. Inhib. hit(s) with Target = 'Cholinesterase' and Ligand = 'BDBM50599167'
TargetCholinesterase(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599167(CHEMBL5195228)
Affinity DataKi:  0.610nMAssay Description:Inhibition of human BChE assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetCholinesterase(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599167(CHEMBL5195228)
Affinity DataIC50:  0.0800nMAssay Description:Inhibition of human BChE using acetylthiocholine iodide or butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599167(CHEMBL5195228)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of horse serum BChE using acetylthiocholine iodide or butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599167(CHEMBL5195228)
Affinity DataKd:  0.370nMAssay Description:Binding affinity to human BChE assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed