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Found 2 Enz. Inhib. hit(s) with Target = 'Cyclin-K/Cyclin-dependent kinase 12' and Ligand = 'BDBM572068'
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572068((R)-N-(4-(3-((7- (methylsulfonyl)quinazolin-2- yl)...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the protein kinase. All kinase assays ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572068((R)-N-(4-(3-((7- (methylsulfonyl)quinazolin-2- yl)...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent