TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataIC50: 0.700nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataIC50: 90nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataIC50: 100nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataIC50: 100nMAssay Description:Binding affinity to CDK2More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataIC50: 100nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataIC50: 220nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataIC50: 400nMAssay Description:Inhibition of CDK2 (unknown origin) after 3 hrs by kinase-glo luminescent assay relative to controlMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataIC50: 430nMAssay Description:Inhibition of human CDK2 using TMB as substrate preincubated for 210 mins followed by substrate addition and measured after 15 to 25 mins by spectrop...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataIC50: 600nMAssay Description:Inhibition of Cyclin-dependent kinase 2 (CDK2/cyclin A)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataIC50: 700nMAssay Description:Inhibition of CDK2/Cyclin A (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataIC50: 700nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataIC50: 700nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataIC50: 700nMAssay Description:Inhibition of CDK2 (unknown origin) in baculovirus infected Sf9 insect cell extract using histone H1 as substrate incubated for 10 mins in presence o...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataKd: 2.90E+3nMAssay Description:Average Binding Constant for CDK2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataKd: 3.40E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataKd: 3.40E+3nMAssay Description:Binding constant for full-length CDK2More data for this Ligand-Target Pair