Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'D(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor' and Ligand = 'BDBM50366495'
LigandChemical structure of BindingDB Monomer ID 50366495BDBM50366495(CHEMBL1255588 | (+)butaclamol)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]- spiperone radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50366495BDBM50366495(CHEMBL1255588 | (+)butaclamol)
Affinity DataIC50: 2nMAssay Description:Concentration inhibiting the specific binding of [3H]spiroperidol by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50366495BDBM50366495(CHEMBL1255588 | (+)butaclamol)
Affinity DataIC50: 13nMAssay Description:Inhibition of [3H]spiroperidol binding to rat striatal membrane using 0.5 nM ligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50366495BDBM50366495(CHEMBL1255588 | (+)butaclamol)
Affinity DataIC50: 50nMAssay Description:The IC50 value was reported as apparent, since [3H]NCA was purported to be irreversible. Result indicates the mean of two separate experiments, each ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed