Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM50021770'
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021770(CHEMBL3298895)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021770(CHEMBL3298895)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human D2L receptor expressed in FlpIn CHO cells assessed as induction of ERK1/2 phosphorylation by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021770(CHEMBL3298895)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at human D2L receptor expressed in FlpIn CHO cells assessed as inhibition of forskolin-stimulated cAMP production treated for 30 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed