Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM50088341'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50088341(11-methyl-11,21-diazatetracyclo[12.7.0.0^{3,8}.0^{...)
Affinity DataKi:  6nMAssay Description:Binding affinity against Dopamine receptor D2 of rat striatal mambranes using [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50088341(11-methyl-11,21-diazatetracyclo[12.7.0.0^{3,8}.0^{...)
Affinity DataKi:  19nMAssay Description:Inhibition of D2L dopamine receptor in HEK 293 cells by intracellular calcium assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50088341(11-methyl-11,21-diazatetracyclo[12.7.0.0^{3,8}.0^{...)
Affinity DataKi:  19nMAssay Description:Activity at human D2L dopamine receptor expressed in HEK293 cells by calcium fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50088341(11-methyl-11,21-diazatetracyclo[12.7.0.0^{3,8}.0^{...)
Affinity DataKi:  41.7nMAssay Description:Displacement of [3H]SCH23390 from human cloned dopamine D2L receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50088341(11-methyl-11,21-diazatetracyclo[12.7.0.0^{3,8}.0^{...)
Affinity DataKi:  44.5nMAssay Description:Displacement of [3H]spiperone from human D2L dopamine receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50088341(11-methyl-11,21-diazatetracyclo[12.7.0.0^{3,8}.0^{...)
Affinity DataKi:  44.5nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50088341(11-methyl-11,21-diazatetracyclo[12.7.0.0^{3,8}.0^{...)
Affinity DataKi:  44.7nMAssay Description:Displacement of [3H]spiperone from D2L dopamine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed