Affinity DataKi: 1.80nMAssay Description:Binding Affinity on high Affinity Site of Bovine dopamine receptor D2. Tested for ability to displace the radioligand [3H]pramipexole was testedMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]-quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-raclopride from high-affinity state of human dopamine D2L receptor (443 amino acids) expressed in LTK deficient mouse fibroblast...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Toronto
Curated by PDSP Ki Database
University of Toronto
Curated by PDSP Ki Database
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]spiperone from human dopamine D2 receptor at high affinity state expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]-NPA from dopamine D2L receptor (unknown origin) expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 8.70nMAssay Description:Displacement of [3H]7-OH-DPAT from human D2 receptor transfected in HEK293 cells measured after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding Affinity was tested on high Affinity Site of Bovine Dopamine D2 Receptor. Tested for ability to displace the radioligand [3H]spiperone was te...More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, high affinity siteMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Toronto
Curated by PDSP Ki Database
University of Toronto
Curated by PDSP Ki Database
Affinity DataKi: 15nMAssay Description:In vitro affinity against Dopamine receptor D2 using [3H]DP-5,6-ADTN radioligand in rat striatal homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-(R)-(+)-7-OH-DPAT from human dopamine D2 receptor expressed in HEK293 cell membranes after 90 mins by micro beta scintillation c...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding Affinity on High Affinity Site of Dopamine receptor D2SMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity on High Affinity Site of Dopamine receptor D2LMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H]-iodosulpiride from cloned human dopamine D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:High binding affinity of the compound for dopamine D-2 receptor from bovine anterior pitutary membrane, using radioligand [3H]-spiroperidolMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Binding Affinity was tested on relative proportion of High Affinity Site of Dopamine receptor D2SMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Binding Affinity was tested on relative proportion of High Affinity Site of Dopamine receptor D2LMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Displacement of [3H]spiperone from human D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Toronto
Curated by PDSP Ki Database
University of Toronto
Curated by PDSP Ki Database
Affinity DataKi: 51nMAssay Description:Binding Affinity was tested on relative proportion of high Affinity Site of Bovine dopamine receptor D2. Tested for ability to displace the radioliga...More data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Displacement of [3H]-iodosulpiride from recombinant high-affinity state of human dopamine D2L receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Toronto
Curated by PDSP Ki Database
University of Toronto
Curated by PDSP Ki Database
Affinity DataKi: 105nMAssay Description:Binding affinity against Dopamine receptor D2 in rat striatal membranes using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Displacement of [3H]spiperone from human dopamine D2short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Displacement of [3H]spiperone from human dopamine D2long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Toronto
Curated by PDSP Ki Database
University of Toronto
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Toronto
Curated by PDSP Ki Database
University of Toronto
Curated by PDSP Ki Database
Affinity DataKi: 197nMAssay Description:Displacement of [3H]raclopride from rat dopamine D2short receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Toronto
Curated by PDSP Ki Database
University of Toronto
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Toronto
Curated by PDSP Ki Database
University of Toronto
Curated by PDSP Ki Database
Affinity DataKi: 231nMAssay Description:Displacement of [3H]spiperone from high-affinity state of human dopamine D2L receptor transfected in HEK293 cells after 2 hrs by scintillation counti...More data for this Ligand-Target Pair
Affinity DataKi: 231nMAssay Description:Displacement of [3H]spiperone from high-affinity state of human dopamine D2L receptor transfected in HEK293 cells after 2 hrs by scintillation counti...More data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 using [3H]spiperone as radioligand transfected in HEK cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Toronto
Curated by PDSP Ki Database
University of Toronto
Curated by PDSP Ki Database
Affinity DataKi: 296nMAssay Description:Inhibitory constant against binding of [125I]- IBZM to rat striatal membraneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Toronto
Curated by PDSP Ki Database
University of Toronto
Curated by PDSP Ki Database
Affinity DataKi: 360nMAssay Description:Displacement of [3H]spiperone from human D2short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 422nMAssay Description:Displacement of [3H]YM-09151-2 from human dopamine D2 receptor expressed in CHOp cellsMore data for this Ligand-Target Pair
Affinity DataKi: 450nMAssay Description:Displacement of [3H]spiperone from human D2long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Toronto
Curated by PDSP Ki Database
University of Toronto
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Toronto
Curated by PDSP Ki Database
University of Toronto
Curated by PDSP Ki Database
Affinity DataKi: 572nMAssay Description:Inhibition of [3H]-raclopride binding to Dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Toronto
Curated by PDSP Ki Database
University of Toronto
Curated by PDSP Ki Database
Affinity DataKi: 617nMAssay Description:Tested for binding affinity against Dopamine receptor D2 like from bovine striatum membranes by using [3H]YM-09151-2 radioligandMore data for this Ligand-Target Pair