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Found 3 Enz. Inhib. hit(s) with Target = 'D(3) dopamine receptor' and Ligand = 'BDBM50016462'
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50016462(CHEMBL3265067)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]R-(+)-7-OHDPAT from dopamine D3 receptor in Sprague-Dawley rat ventral striatum after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50016462(CHEMBL3265067)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50016462(CHEMBL3265067)
Affinity DataIC50:  327nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in human U2OS cells assessed as inhibition of pramipexole-stimulated beta-arrestin recrui...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed