Affinity DataKi: 5.20nMAssay Description:Binding Affinity was tested on the high affinity site of Dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding Affinity was tested on relative proportion of High Affinity Site of Dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Displacement of [3H]spiperone from human wild type D3 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Dissociation constant of compound on one-site model Human Dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataKi: 590nMAssay Description:Binding Affinity was tested on low Affinity Site of Dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataKi: 720nMAssay Description:Binding Affinity was determined in the presence of 100 micro M Gpp(NH)p for decoupling of the ternary complex of Compound to Dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataEC50: 4.40nMAssay Description:Intrinsic activity at human D3 receptor expressed in CHO dhfr- cells by [3H]thymidine incorporation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.70nMAssay Description:Intrinsic activity at human D3 receptor expressed in CHO dhfr- cells assessed as inhibition of forskolin-induced cAMP releaseMore data for this Ligand-Target Pair