Found 3 Enz. Inhib. hit(s) with Target = 'DNA (cytosine-5)-methyltransferase 3A' and Ligand = 'BDBM50430056' TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
M. V. Lomonosov Moscow State University
Curated by ChEMBL
M. V. Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of human C-terminal DNMT3A (623 to 908 residues) using 5'-biotin labeled oligonucleotide as substrate measured after 1 hrMore data for this Ligand-Target Pair
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
M. V. Lomonosov Moscow State University
Curated by ChEMBL
M. V. Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of His6-tagged human recombinant DNMT3a expressed in insect Sf9 cells assessed as reduction in DNA methyltransferase activity using 5'-bio...More data for this Ligand-Target Pair
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
M. V. Lomonosov Moscow State University
Curated by ChEMBL
M. V. Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataEC50: 900nMAssay Description:Inhibition of human C-terminal DNMT3A after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
