Found 1 Enz. Inhib. hit(s) with Target = 'DNA (cytosine-5)-methyltransferase 3A' and Ligand = 'BDBM50544059'
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
M. V. Lomonosov Moscow State University
Curated by ChEMBL
M. V. Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Binding affinity to DNMT3A catalytic domain (unknown origin) assessed as inhibition of enzyme-mediated DNA methylation preincubated for 1 hr followed...More data for this Ligand-Target Pair