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Found 1 Enz. Inhib. hit(s) with Target = 'DNA (cytosine-5)-methyltransferase 3A' and Ligand = 'BDBM50544059'
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
M. V. Lomonosov Moscow State University

Curated by ChEMBL
LigandPNGBDBM50544059(CHEMBL4171551)
Affinity DataIC50:  6.00E+3nMAssay Description:Binding affinity to DNMT3A catalytic domain (unknown origin) assessed as inhibition of enzyme-mediated DNA methylation preincubated for 1 hr followed...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed