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Found 4 Enz. Inhib. hit(s) with Target = 'DNA polymerase catalytic subunit' and Ligand = 'BDBM50172517'
TargetDNA polymerase catalytic subunit(Varicella-zoster virus (strain Dumas) (HHV-3) (Hum...)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50172517(4-Hydroxy-6-(3-hydroxy-propyl)-quinoline-3-carboxy...)
Affinity DataIC50:  70nMpH: 7.5Assay Description:Inhibition of Varicella-Zoster virus DNA polymerase (95 uL) activity in a solution containing 6.4 mM HEPES (pH 7.5), incubation for 12 minutes at 26 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase catalytic subunit(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50172517(4-Hydroxy-6-(3-hydroxy-propyl)-quinoline-3-carboxy...)
Affinity DataIC50:  300nMpH: 7.5Assay Description:Inhibition of herpes simplex virus type 1 DNA polymerase (95 uL) activity in a solution containing 6.4 mM HEPES (pH 7.5), incubation for 12 minutes a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase catalytic subunit(Human cytomegalovirus (HCMV strain AD169) )
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50172517(4-Hydroxy-6-(3-hydroxy-propyl)-quinoline-3-carboxy...)
Affinity DataIC50:  400nMpH: 7.5Assay Description:Inhibition of human cytomegalovirus DNA polymerase (95 uL) activity in a solution containing 6.4 mM HEPES (pH 7.5), incubation for 12 minutes at 26 d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase catalytic subunit(Varicella-zoster virus (strain Dumas) (HHV-3) (Hum...)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50172517(4-Hydroxy-6-(3-hydroxy-propyl)-quinoline-3-carboxy...)
Affinity DataIC50: >4.00E+4nMpH: 7.5Assay Description:Inhibition of Varicella-Zoster virus DNA polymerase (95 uL) activity in a solution containing 6.4 mM HEPES (pH 7.5), incubation for 12 minutes at 26 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed