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Found 2 Enz. Inhib. hit(s) with Target = 'DNA-(apurinic or apyrimidinic site) endonuclease' and Ligand = 'BDBM50530043'
TargetDNA-(apurinic or apyrimidinic site) endonuclease(Homo sapiens (Human))
Boston University

Curated by ChEMBL
LigandPNGBDBM50530043(CHEMBL4458126)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of full length human APE1 assessed as reduction in endonuclease activity by measuring DNA cleavage of abasic sites using 6-FAM labelled tw...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA-(apurinic or apyrimidinic site) endonuclease(Homo sapiens (Human))
Boston University

Curated by ChEMBL
LigandPNGBDBM50530043(CHEMBL4458126)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of full length human APE1 assessed as reduction in endonuclease activity by measuring DNA cleavage of abasic sites using 6-FAM labelled tw...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed