Found 1 Enz. Inhib. hit(s) with Target = 'DNA-(apurinic or apyrimidinic site) endonuclease' and Ligand = 'BDBM58109'
TargetDNA-(apurinic or apyrimidinic site) endonuclease(Homo sapiens (Human))
Russian Academy Of Sciences
Curated by ChEMBL
Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of nuclease activity of APE1 in human glioblastoma cells assessed as reduction in AP site DNA cleavageMore data for this Ligand-Target Pair