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Found 1 Enz. Inhib. hit(s) with Target = 'DNA-dependent protein kinase catalytic subunit/Serine/threonine-protein kinase mTOR' and Ligand = 'BDBM36409'
TargetDNA-dependent protein kinase catalytic subunit/Serine/threonine-protein kinase mTOR(Homo sapiens (Human))
University of California San Francisco

LigandPNGBDBM36409(2-(4-amino-1-isopropyl-1H-pyrazolo[3,4-d]pyrimidin...)
Affinity DataIC50:  410nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair