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Found 6 Enz. Inhib. hit(s) with Target = 'Delta-type opioid receptor' and Ligand = 'BDBM50009185'
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50009185(4-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylami...)
Affinity DataKi:  0.120nMAssay Description:Binding affinity against opioid receptor delta in rats by displacing [3H]-DPDPEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50009185(4-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylami...)
Affinity DataKi:  0.310nMAssay Description:Inhibition of [3H]-DADLE binding to opioid receptor delta in P2 membrane preparation of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50009185(4-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylami...)
Affinity DataKi:  0.410nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50009185(4-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylami...)
Affinity DataIC50:  5.60nMAssay Description:In vitro opioid receptor delta mediated mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50009185(4-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylami...)
Affinity DataIC50:  184nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50009185(4-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylami...)
Affinity DataEC50:  0.331nMAssay Description:Negative logarithm of the molar concentration of delta receptor was determined in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed