Affinity DataKi: 0.199nMAssay Description:Binding affinity to delta opioid receptor in Sprague-Dawley rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 129nMAssay Description:Agonist activity at delta opioid receptor assessed as inhibition of electrically-stimulated mouse vas deferens contractionMore data for this Ligand-Target Pair