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Found 3 Enz. Inhib. hit(s) with Target = 'Deoxycytidine kinase' and Ligand = 'BDBM50031349'
TargetDeoxycytidine kinase(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50031349(CHEMBL3358094)
Affinity DataKi:  6.80nMAssay Description:Apparent inhibition of human dCK by steady-state kinetic assayMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50031349(CHEMBL3358094)
Affinity DataIC50:  7nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of [3H]-dC uptake by scintillation counting analysisMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50031349(CHEMBL3358094)
Affinity DataIC50:  25nMAssay Description:Apparent inhibition of human dCK assessed as phosphorylation activity by spectroscopic NADH-dependent enzyme-coupled assayMore data for this Ligand-Target Pair