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Found 1 Enz. Inhib. hit(s) with Target = 'Diacylglycerol O-acyltransferase 2' and Ligand = 'BDBM530640'
TargetDiacylglycerol O-acyltransferase 2(Homo sapiens (Human))
Merck Sharp &Amp

WIPO
LigandPNGBDBM530640(WO2022076495, EXAMPLE 75a)
Affinity DataIC50:  1.5nMAssay Description:DGAT2 activity was determined by measuring the amount of enzymatic product 13Ci8-triolein (13C-l,2,3-Tri(cis-9-octadecenoyl)glycerol) using the membr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed