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Found 3 Enz. Inhib. hit(s) with Target = 'Dual specificity protein kinase CLK1' and Ligand = 'BDBM50552555'
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Chemveda Life Sciences India

Curated by ChEMBL
LigandPNGBDBM50552555(CHEMBL4783398)
Affinity DataIC50:  11nMAssay Description:Inhibition of recombinant human CLK1 (130 to end residues) using ERMRPRKRQGSVRRRV as substrate incubated for 40 mins in presence of [gamma33P-ATP] by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Chemveda Life Sciences India

Curated by ChEMBL
LigandPNGBDBM50552555(CHEMBL4783398)
Affinity DataIC50:  3.88E+3nMAssay Description:Inhibition of recombinant human CLK1 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scinti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Chemveda Life Sciences India

Curated by ChEMBL
LigandPNGBDBM50552555(CHEMBL4783398)
Affinity DataKd:  112nMAssay Description:Binding affinity to human CLK1 assessed as equilibrium dissociation constant measured upto 240 min by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed