Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Dual specificity tyrosine-phosphorylation-regulated kinase 1B' and Ligand = 'BDBM246384'
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM246384(US9446044, 71)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of human DYRK1B using [33P]-ATP incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM246384(US9446044, 71)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of DYRK1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM246384(US9446044, 71)
Affinity DataIC50:  1.63nMpH: 7.5 T: 2°CAssay Description:The DYRK1A and DYRK1B kinase assays to determine IC50 values were performed by Reaction Biology Corporation using HotSpot technology Worldwide websit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent