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Found 2 Enz. Inhib. hit(s) with Target = 'Ecdysone receptor' and Ligand = 'BDBM50488437'
TargetEcdysone receptor(Bombyx mori)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488437(CHEMBL2286416)
Affinity DataIC50:  1.48E+4nMAssay Description:Antagonist activity at ecdysone receptor in Bombyx mori Bm5 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide challenge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Spodoptera littoralis)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488437(CHEMBL2286416)
Affinity DataIC50:  7.94E+4nMAssay Description:Antagonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells assessed as tebufenozide-induced effect treated 24 hr before tebufenozide...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed