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Found 1 Enz. Inhib. hit(s) with Target = 'Estrogen receptor [298-554,D538G]' and Ligand = 'BDBM521352'
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM521352(5-[4-[(3S)-1-(3- fluoropropyl)pyr- rolidin-3- yl]o...)
Affinity DataIC50:  28nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent