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Found 1 Enz. Inhib. hit(s) with Target = 'Estrogen receptor [298-554,D538G]' and Ligand = 'BDBM521382'
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM521382(4-(2-chloro-4- methyl-phenyl)- 5-[6-[(3S)-1-(3- fl...)
Affinity DataIC50:  13nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent